H7 dihydrochloride
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Hodoodo CAT#: H540189

CAS#: 108930-17-2 (HCl)

Description: H7 is a specific protein kinase C inhibitor and protein kinase G inhibitor, which inhibits superoxide release from human neutrophils (PMN) stimulated with phorbol myristate acetate or synthetic diacylglycerol.


Chemical Structure

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H7 dihydrochloride
CAS# 108930-17-2 (HCl)

Theoretical Analysis

Hodoodo Cat#: H540189
Name: H7 dihydrochloride
CAS#: 108930-17-2 (HCl)
Chemical Formula: C31H42N6O5S
Exact Mass: 0.00
Molecular Weight: 364.285
Elemental Analysis: C, 60.96; H, 6.93; N, 13.76; O, 13.10; S, 5.25

Price and Availability

Size Price Availability Quantity
10mg USD 285 2 Weeks
25mg USD 500 2 Weeks
50mg USD 850 2 Weeks
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Related CAS #: 108930-17-2 (HCl)   84477-87-2 (free base)    

Synonym: H7 dihydrochloride; H7 HCl.

IUPAC/Chemical Name: 5-((2-methylpiperazin-1-yl)sulfonyl)isoquinoline dihydrochloride

InChi Key: OARGPFMFRLLKPF-UHFFFAOYSA-N

InChi Code: InChI=1S/C14H17N3O2S.2ClH/c1-11-9-16-7-8-17(11)20(18,19)14-4-2-3-12-10-15-6-5-13(12)14;;/h2-6,10-11,16H,7-9H2,1H3;2*1H

SMILES Code: O=S(C1=CC=CC2=C1C=CN=C2)(N3C(C)CNCC3)=O.[H]Cl.[H]Cl

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 364.29 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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