R(+)-6-Bromo-APB HBr
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Hodoodo CAT#: H563376

CAS#: 139689-19-3

Description: R(+)-6-Bromo-APB HBr is a potent D1 Dopamine receptor agonist.

Chemical Structure

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R(+)-6-Bromo-APB HBr
CAS# 139689-19-3
Instruction

Theoretical Analysis

Hodoodo Cat#: H563376
Name: R(+)-6-Bromo-APB HBr
CAS#: 139689-19-3
Chemical Formula: C19H21Br2NO2
Exact Mass: 0.00
Molecular Weight: 455.190
Elemental Analysis: C, 50.13; H, 4.65; Br, 35.11; N, 3.08; O, 7.03

Price and Availability

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25mg USD 620 2 weeks
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Synonym: R(+)-6-Bromo-APB hydrobromide; R(+) 6 Bromo APB hydrobromide; R(+)-6-Bromo-APB HBr; R(+) 6 Bromo APB HBr;

IUPAC/Chemical Name: (R)-3-allyl-6-bromo-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol hydrobromide

InChi Key: CTAUBYSSTAODOD-PKLMIRHRSA-N

InChi Code: InChI=1S/C19H20BrNO2.BrH/c1-2-9-21-10-8-14-15(11-17(22)19(23)18(14)20)16(12-21)13-6-4-3-5-7-13;/h2-7,11,16,22-23H,1,8-10,12H2;1H/t16-;/m1./s1

SMILES Code: OC1=C(O)C=C2[C@@H](C3=CC=CC=C3)CN(CC=C)CCC2=C1Br.Br

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.03.00

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 455.19 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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5: Azaryan AV, Clock BJ, Cox BM. Mu opioid receptor mRNA in nucleus accumbens is elevated following dopamine receptor activation. Neurochem Res. 1996 Nov;21(11):1411-5. PubMed PMID: 8947931.