Aminolevulinic acid phosphate

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Hodoodo CAT#: H573886

CAS#: 868074-65-1 (phosphate)

Description: Aminolevulinic acid phosphate is a topically administered metabolic precursor of protoporphyrin IX. After topical administration, aminolevulinic acid (ALA) is converted to protoporphyrin IX (PpIX) which is a photosensitizer. When the proper wavelength of light activates protoporphyrin IX, singlet oxygen is produced, resulting in a local cytotoxic effect.


Chemical Structure

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Aminolevulinic acid phosphate
CAS# 868074-65-1 (phosphate)

Theoretical Analysis

Hodoodo Cat#: H573886
Name: Aminolevulinic acid phosphate
CAS#: 868074-65-1 (phosphate)
Chemical Formula: C5H12NO7P
Exact Mass: 229.04
Molecular Weight: 229.120
Elemental Analysis: C, 26.21; H, 5.28; N, 6.11; O, 48.88; P, 13.52

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @hodoodo.com or click below button.
Note: Price will be listed if it is available in the future.

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Related CAS #: 5451-09-2 (HCl)   106-60-5 (free)   868074-65-1 (phosphate)  

Synonym: 5-Aminolevulinic acid phosphate, Aminolevulinic acid phosphate, delta-Aminolevulinic acid phosphate

IUPAC/Chemical Name: Pentanoic acid, 5-amino-4-oxo-, phosphate (1:1)

InChi Key: XWNWBYZHOAIHTK-UHFFFAOYSA-N

InChi Code: 1S/C5H9NO3.H3O4P/c6-3-4(7)1-2-5(8)9;1-5(2,3)4/h1-3,6H2,(H,8,9);(H3,1,2,3,4)

SMILES Code: C(CC(=O)O)C(=O)CN.OP(=O)(O)O

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 229.12 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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