Formylmelphalan
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    WARNING: This product is for research use only, not for human or veterinary use.

Hodoodo CAT#: H100382

CAS#: 7789-59-5

Description: Formylmelphalan was approved in China for treating cancer. Formylmelphalan is an alkylating agents, which could cross-link DNA.


Chemical Structure

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Formylmelphalan
CAS# 7789-59-5

Theoretical Analysis

Hodoodo Cat#: H100382
Name: Formylmelphalan
CAS#: 7789-59-5
Chemical Formula: C14H18Cl2N2O3
Exact Mass: 332.07
Molecular Weight: 333.210
Elemental Analysis: C, 50.46; H, 5.44; Cl, 21.28; N, 8.41; O, 14.40

Price and Availability

Size Price Availability Quantity
5g USD 350 2 Weeks
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Synonym: NFormylmelphalan; NFormylLsarcolysin; NFormylLpsarcolysin; CB 3208; NSC 37024; NSC37024; LS15879.

IUPAC/Chemical Name: 3-[4-[bis(2-chloroethyl)amino]phenyl]-2-formamidopropanoic acid

InChi Key: ZPOLNCDBPYJDSE-UHFFFAOYSA-N

InChi Code: InChI=1S/C14H18Cl2N2O3/c15-5-7-18(8-6-16)12-3-1-11(2-4-12)9-13(14(20)21)17-10-19/h1-4,10,13H,5-9H2,(H,17,19)(H,20,21)

SMILES Code: O=C(O)C(NC=O)CC1=CC=C(N(CCCl)CCCl)C=C1

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:        

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 333.21 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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