Azatadine Maleate
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Hodoodo CAT#: H317301

CAS#: 3978-86-7

Description: Azatadine dimaleate is an antihistamine and anticholinergic inhibitor. It is used for treating allergic rhinitis and chronic urticaria.

Chemical Structure

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Azatadine Maleate
CAS# 3978-86-7
Instruction

Theoretical Analysis

Hodoodo Cat#: H317301
Name: Azatadine Maleate
CAS#: 3978-86-7
Chemical Formula: C28H30N2O8
Exact Mass: 522.20
Molecular Weight: 522.550
Elemental Analysis: C, 64.36; H, 5.79; N, 5.36; O, 24.49

Price and Availability

Size Price Availability Quantity
20mg USD 210 2 Weeks
50mg USD 280 2 Weeks
250mg USD 380 2 Weeks
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Synonym: Azatadine Maleate; azatadine; azatadine maleate; Idulamine; Idulian; Juste brand of azatadine maleate; Key brand of azatadine maleate; Lergocil; Optimine; Schering brand of azatadine maleate; Schering-Plough brand of azatadine maleate; Zadine

IUPAC/Chemical Name: 6,11-Dihydro-11-(1-methylpiperidin-4-ylidene)-5H-benzo[5,6]cyclohepta[1,2-b]pyridine dimaleate

InChi Key: SGHXFFAHXTZRQM-SPIKMXEPSA-N

InChi Code: InChI=1S/C20H22N2.2C4H4O4/c1-22-13-10-16(11-14-22)19-18-7-3-2-5-15(18)8-9-17-6-4-12-21-20(17)19;2*5-3(6)1-2-4(7)8/h2-7,12H,8-11,13-14H2,1H3;2*1-2H,(H,5,6)(H,7,8)/b;2*2-1-

SMILES Code: CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=CC=CN=C4\2.O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 522.55 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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18: Kaplan AP. Exercise-induced hives. J Allergy Clin Immunol. 1984 May;73(5 Pt 2):704-7. doi: 10.1016/0091-6749(84)90310-5. PMID: 6371106.


19: Wilson JD, Hillas JL, Somerfield SD. Azatadine maleate (Zadine): evaluation in the management of allergic rhinitis. N Z Med J. 1981 Aug 12;94(689):79-81. PMID: 7024868.


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