Elvitegravir

CAT#: H314218

CAS#:


Description: Elvitegravir, also known as GS-9137 ans EVG, is an integrase inhibitor used to treat HIV infection. The drug gained approval by the U.S. Food and Drug Administration on August 27, 2012 for use in adult patients starting HIV treatment for the first time as part of the fixed dose combination known as Stribild.

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Synthetic Routes

Elvitegravir - Synthetic Route 1

Elvitegravir route01

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Elvitegravir - Synthetic Route 2

Elvitegravir route02

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Elvitegravir - Synthetic Route 3

Elvitegravir route03

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Elvitegravir - Synthetic Route 4

Elvitegravir route04

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Elvitegravir - Synthetic Route 5

Elvitegravir route05

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Elvitegravir - Synthetic Route 6

Elvitegravir route06

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Elvitegravir - Synthetic Route 7

Elvitegravir route07

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Elvitegravir - Synthetic Route 8

Elvitegravir route08

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Elvitegravir - Synthetic Route 9

Elvitegravir route09

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Elvitegravir - Synthetic Route 10

Elvitegravir route010

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Elvitegravir - Synthetic Route 11

Elvitegravir route011

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Ma, Shuai; Zhao, Jun; Du, Weihong; Cao, Shenghua. Synthesis of elvitegravir. Zhongguo Yiyao Gongye Zazhi. Sichuan Industrial Institute of Antibiotics. China National Pharmaceutical Group Co. Chengdu, Sichuan Province, Peop. Rep. China 610052. Volume 45. Issue 1. Pages 5-8. 2014.