DC_M01_7

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Hodoodo CAT#: H130582

CAS#: DC_M01_7

Description: DC_M01_7 is a novel inhibitor of human histone acetyltransferase KAT8 (also known as MOF or MYST1) with an IC50 value of 6 μM. It significantly inhibits HCT116 cells proliferation and also inhibiting histone 4 lysine 16 acetylation in HCT116 cells.

Chemical Structure

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DC_M01_7
CAS# DC_M01_7
Instruction

Theoretical Analysis

Hodoodo Cat#: H130582
Name: DC_M01_7
CAS#: DC_M01_7
Chemical Formula: C19H20N2O2S2
Exact Mass: 372.10
Molecular Weight: 372.500
Elemental Analysis: C, 61.26; H, 5.41; N, 7.52; O, 8.59; S, 17.21

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @hodoodo.com or click below button.
Note: Price will be listed if it is available in the future.

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Synonym: DC M01 7, DC-M01-7, DCM017, DC M01-7, DC_M01 7, DC M01_7

IUPAC/Chemical Name: (E)-4-(2-(Benzo[d]thiazol-2-yl)vinyl)-N,N-diethylbenzenesulfonamide

InChi Key: IYTCMWSUAKFEFW-SDNWHVSQSA-N

InChi Code: InChI=1S/C19H20N2O2S2/c1-3-21(4-2)25(22,23)16-12-9-15(10-13-16)11-14-19-20-17-7-5-6-8-18(17)24-19/h5-14H,3-4H2,1-2H3/b14-11+

SMILES Code: O=S(C(C=C1)=CC=C1/C=C/C(S2)=NC3=C2C=CC=C3)(N(CC)CC)=O

Appearance: To be determined

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: To be determined

Shelf Life: >2 years if stored properly

Drug Formulation: To be determined

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 372.50 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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1. Zhang R, Wang J, Zhao L, Liu S, Du D, Ding H, Chen S, Yue L, Liu YC, Zhang C, Liu H, Luo C. Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening. Eur J Med Chem. 2018 Sep 5;157:867-876. doi: 10.1016/j.ejmech.2018.08.026. Epub 2018 Aug 17. PMID: 30145373.