WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H532163
CAS#: 2829282-00-8
Description: LY367385 is a selective mGlu1a receptor antagonist, with an IC50 value of 8.8 μM for blockade of quisqualate-induced phosphoinositide hydrolysis.
Hodoodo Cat#: H532163
Name: LY367385 HCl
CAS#: 2829282-00-8
Chemical Formula: C10H12ClNO4
Exact Mass: 209.07
Molecular Weight: 245.659
Elemental Analysis: C, 48.89; H, 4.92; Cl, 14.43; N, 5.70; O, 26.05
Related CAS #: 198419-91-9 (free base) LY367385 HCl,
Synonym: LY367385; LY 367385; LY-367385; LY367385 HCl; LY367385 hydrochloride
IUPAC/Chemical Name: 4-[(1S)-1-amino-2-hydroxy-2-oxoethyl]-3-methylbenzoic acid hydrochloride
InChi Key: IGKQWSUZDKTEPR-QRPNPIFTSA-N
InChi Code: InChI=1S/C10H11NO4.ClH/c1-5-4-6(9(12)13)2-3-7(5)8(11)10(14)15;/h2-4,8H,11H2,1H3,(H,12,13)(H,14,15);1H/t8-;/m0./s1
SMILES Code: O=C(O)C1=CC=C([C@H](N)C(O)=O)C(C)=C1.[H]Cl
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
More Info:
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The following data is based on the product molecular weight 245.66 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
Formulation protocol: | |
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In vivo protocol: |