WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H532266
CAS#: 70460-45-6
Description: MRS1067 is an A3 adenosine receptor antagonist.
Hodoodo Cat#: H532266
Name: MRS1067
CAS#: 70460-45-6
Chemical Formula: C19H16Cl2O3
Exact Mass: 362.05
Molecular Weight: 363.230
Elemental Analysis: C, 62.83; H, 4.44; Cl, 19.52; O, 13.21
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Synonym: MRS1067 ; MRS 1067 ; MRS-1067.
IUPAC/Chemical Name: 3,6-dichloro-2-(4-methyl-2-propan-2-yloxyphenyl)chromen-4-one
InChi Key: PWGZOUCWGRTPSM-UHFFFAOYSA-N
InChi Code: InChI=1S/C19H16Cl2O3/c1-10(2)23-16-8-11(3)4-6-13(16)19-17(21)18(22)14-9-12(20)5-7-15(14)24-19/h4-10H,1-3H3
SMILES Code: O=C1C(Cl)=C(C2=CC=C(C)C=C2OC(C)C)OC3=C1C=C(Cl)C=C3
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
More Info:
Biological target: | |
In vitro activity: | |
In vivo activity: |
The following data is based on the product molecular weight 363.23 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
Formulation protocol: | |
In vitro protocol: | |
In vivo protocol: |
1: Jacobson KA, Park KS, Jiang JL, Kim YC, Olah ME, Stiles GL, Ji XD. Pharmacological characterization of novel A3 adenosine receptor-selective antagonists. Neuropharmacology. 1997 Sep;36(9):1157-65. PubMed PMID: 9364471; PubMed Central PMCID: PMC3433714.