Pentamidine
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Hodoodo CAT#: H527056

CAS#: 100-33-4

Description: Pentamidine is an antiprotozoal and antifungal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor groove of DNA, thereby interfering with DNA replication.

Chemical Structure

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Pentamidine
CAS# 100-33-4
Instruction

Theoretical Analysis

Hodoodo Cat#: H527056
Name: Pentamidine
CAS#: 100-33-4
Chemical Formula: C19H24N4O2
Exact Mass: 340.19
Molecular Weight: 340.427
Elemental Analysis: C, 67.04; H, 7.11; N, 16.46; O, 9.40

Price and Availability

Size Price Availability Quantity
100mg USD 250
250mg USD 440
500mg USD 750
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Synonym: Pentamidine

IUPAC/Chemical Name: 4-[5-(4-Carbamimidoylphenoxy)pentoxy]benzenecarboximidamide

InChi Key: XDRYMKDFEDOLFX-UHFFFAOYSA-N

InChi Code: InChI=1S/C19H24N4O2/c20-18(21)14-4-8-16(9-5-14)24-12-2-1-3-13-25-17-10-6-15(7-11-17)19(22)23/h4-11H,1-3,12-13H2,(H3,20,21)(H3,22,23)

SMILES Code: N=C(C1=CC=C(OCCCCCOC2=CC=C(C(N)=N)C=C2)C=C1)N

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 340.43 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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