KG-501
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    WARNING: This product is for research use only, not for human or veterinary use.

Hodoodo CAT#: H562626

CAS#: 18228-17-6

Description: KG-501 is a cAMP response element-binding protein (CREB) inhibitor.

Chemical Structure

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KG-501
CAS# 18228-17-6
Instruction

Theoretical Analysis

Hodoodo Cat#: H562626
Name: KG-501
CAS#: 18228-17-6
Chemical Formula: C17H13ClNO5P
Exact Mass: 377.02
Molecular Weight: 377.710
Elemental Analysis: C, 54.06; H, 3.47; Cl, 9.39; N, 3.71; O, 21.18; P, 8.20

Price and Availability

Size Price Availability Quantity
200mg USD 450 2 Weeks
500mg USD 850 2 Weeks
1g USD 1450 2 Weeks
2g USD 2450 2 Weeks
5g USD 5450 2 Weeks
Bulk inquiry

Synonym: KG-501; KG 501; KG501;

IUPAC/Chemical Name: N-(4-Chlorophenyl)-3-(phosphonooxy)naphthalene-2-carboxamide

InChi Key: RQAQWBFHPMSXKR-UHFFFAOYSA-N

InChi Code: InChI=1S/C17H13ClNO5P/c18-13-5-7-14(8-6-13)19-17(20)15-9-11-3-1-2-4-12(11)10-16(15)24-25(21,22)23/h1-10H,(H,19,20)(H2,21,22,23)

SMILES Code: O=C(C1=C(OP(O)(O)=O)C=C2C=CC=CC2=C1)NC3=CC=C(Cl)C=C3

Appearance: Solid powder

Purity: >97% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 377.71 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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