WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H598089
CAS#: 132472-84-5
Description: QF-Erp7 is a novel quenched fluorescence substrate structurally related to enkephalin.
Hodoodo Cat#: H598089
Name: QF-Erp7
CAS#: 132472-84-5
Chemical Formula: C51H74N18O12
Exact Mass: 1,130.57
Molecular Weight: 1,131.260
Elemental Analysis: C, 54.15; H, 6.59; N, 22.29; O, 16.97
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Synonym: QF-Erp7; QF Erp7; QFErp7; Abz-G-G-F-L-R-R-V-eddn;
IUPAC/Chemical Name: 2-amino-N-((6S,9S,12S,15S)-1-amino-6-(((S)-1-amino-3-methyl-1-oxobutan-2-yl)(2-((2,4-dinitrophenyl)amino)ethyl)carbamoyl)-15-benzyl-9-(3-guanidinopropyl)-1-imino-12-isobutyl-8,11,14,17,20-pentaoxo-2,7,10,13,16,19-hexaazahenicosan-21-yl)benzamide
InChi Key: JDYFMQPAPMPKCG-WWFQFRPWSA-N
InChi Code: InChI=1S/C51H74N18O12/c1-29(2)24-38(66-48(76)39(25-31-12-6-5-7-13-31)63-42(71)28-61-41(70)27-62-45(73)33-14-8-9-15-34(33)52)47(75)64-36(16-10-20-59-50(54)55)46(74)65-37(17-11-21-60-51(56)57)49(77)67(43(30(3)4)44(53)72)23-22-58-35-19-18-32(68(78)79)26-40(35)69(80)81/h5-9,12-15,18-19,26,29-30,36-39,43,58H,10-11,16-17,20-25,27-28,52H2,1-4H3,(H2,53,72)(H,61,70)(H,62,73)(H,63,71)(H,64,75)(H,65,74)(H,66,76)(H4,54,55,59)(H4,56,57,60)/t36-,37-,38-,39-,43-/m0/s1
SMILES Code: CC(C)[C@@H](C(N)=O)N(C([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@H](CC1=CC=CC=C1)NC(CNC(CNC(C2=CC=CC=C2N)=O)=O)=O)=O)=O)=O)=O)CCNC3=CC=C([N+]([O-])=O)C=C3[N+]([O-])=O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.03.00
More Info:
Biological target: | |
In vitro activity: | |
In vivo activity: |
The following data is based on the product molecular weight 1,131.26 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
Formulation protocol: | |
In vitro protocol: | |
In vivo protocol: |
1: Juliano L, Chagas JR, Hirata IY, Carmona E, Sucupira M, Oliveira ES, Oliveira EB, Camargo AC. A selective assay for endooligopeptidase A based on the cleavage of fluorogenic substrate structurally related to enkephalin. Biochem Biophys Res Commun. 1990 Dec 14;173(2):647-52. PubMed PMID: 2260976.
2: Ferro ES, Tambourgy DV, Abreu PA, Camargo AC, Raw I, Ho PL. Characterization of an endooligopeptidase A-like protein in PC12 cells: activity modulation by cAMP but not by basic fibroblast growth factor. J Cell Biochem. 1995 Feb;57(2):311-20. PubMed PMID: 7759568.