WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H462869
CAS#: 33089-74-6
Description: U-40481 reduced the rate of both 45Ca uptake and norepinephrine-stimulated 45Ca uptake into deadventitiated rabbit aorta strips and reduced NE-stimulated efflux from 45Ca-loaded, superfused aorta strips.
Hodoodo Cat#: H462869
Name: U-40481
CAS#: 33089-74-6
Chemical Formula: C10H14N2
Exact Mass: 162.12
Molecular Weight: 162.236
Elemental Analysis: C, 74.03; H, 8.70; N, 17.27
This product is not in stock, which may be available by custom synthesis.
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Note: Price will be listed if it is available in the future.
Synonym: U-40481; U 40481A; NSC363957; NSC-363957; NSC 363957;
IUPAC/Chemical Name: (E)-N-(2,4-dimethylphenyl)-N'-methylformimidamide
InChi Key: JIIOLEGNERQDIP-UHFFFAOYSA-N
InChi Code: InChI=1S/C10H14N2/c1-8-4-5-10(9(2)6-8)12-7-11-3/h4-7H,1-3H3,(H,11,12)
SMILES Code: C/N=C/Nc1c(C)cc(C)cc1
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
More Info:
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| In vitro activity: | |
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The following data is based on the product molecular weight 162.24 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
| Formulation protocol: | |
| In vitro protocol: | |
| In vivo protocol: |
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