WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H471094
CAS#: 1421349-19-0
Description: PF-06412154 HCl is a glucagon receptor antagonist.
Hodoodo Cat#: H471094
Name: PF-06412154 HCl
CAS#: 1421349-19-0
Chemical Formula: C24H28ClN3O3
Exact Mass: 0.00
Molecular Weight: 441.960
Elemental Analysis: C, 65.22; H, 6.39; Cl, 8.02; N, 9.51; O, 10.86
Synonym: PF-06412154 HCl; PF06412154 HCl; PF 06412154 HCl
IUPAC/Chemical Name: (R)-3-(4-(1-((3-methylquinolin-2-yl)amino)butyl)benzamido)propanoic acid hydrochloride
InChi Key: BTOHFLWOXYLUQK-VEIFNGETSA-N
InChi Code: InChI=1S/C24H27N3O3.ClH/c1-3-6-20(26-23-16(2)15-19-7-4-5-8-21(19)27-23)17-9-11-18(12-10-17)24(30)25-14-13-22(28)29;/h4-5,7-12,15,20H,3,6,13-14H2,1-2H3,(H,25,30)(H,26,27)(H,28,29);1H/t20-;/m1./s1
SMILES Code: [H]Cl.OC(CCNC(C1=CC=C(C=C1)[C@@H](CCC)NC2=C(C=C3C=CC=CC3=N2)C)=O)=O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: To be determined
Shelf Life: >2 years if stored properly
Drug Formulation: To be determined
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
More Info:
Biological target: | |
In vitro activity: | |
In vivo activity: |
The following data is based on the product molecular weight 441.96 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
Formulation protocol: | |
In vitro protocol: | |
In vivo protocol: |