WARNING: This product is for research use only, not for human or veterinary use.
Hodoodo CAT#: H524806
CAS#: 86329-06-8
Description: CP 59430 is an azide analog of prazosin, a highly selective alpha 1-adrenergic receptor antagonist.
Hodoodo Cat#: H524806
Name: CP 59430
CAS#: 86329-06-8
Chemical Formula: C21H22N8O3
Exact Mass: 0.00
Molecular Weight: 434.450
Elemental Analysis: C, 58.06; H, 5.10; N, 25.79; O, 11.05
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Synonym: CP 59430; CP59430; CP-59430.
IUPAC/Chemical Name: 2-(4-(4-Azidobenzoyl)piperazin-1-yl)-4-amino-6,7-dimethoxyquinazoline
InChi Key: XHCZPSMUDVXSPQ-UHFFFAOYSA-N
InChi Code: InChI=1S/C21H22N8O3/c1-31-17-11-15-16(12-18(17)32-2)24-21(25-19(15)22)29-9-7-28(8-10-29)20(30)13-3-5-14(6-4-13)26-27-23/h3-6,11-12H,7-10H2,1-2H3,(H2,22,24,25)
SMILES Code: COc1cc2c(cc1OC)nc(nc2N)N3CCN(CC3)C(=O)c4ccc(cc4)N=[N+]=[N-]
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
More Info:
Biological target: | |
In vitro activity: | |
In vivo activity: |
The following data is based on the product molecular weight 434.45 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
Formulation protocol: | |
In vitro protocol: | |
In vivo protocol: |
1: Hess HJ, Graham RM, Homcy CJ. Photoaffinity label for the alpha 1-adrenergic receptor: synthesis and effects on membrane and affinity-purified receptors. Proc Natl Acad Sci U S A. 1983 Apr;80(8):2102-6. PubMed PMID: 6300894; PubMed Central PMCID: PMC393765.